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-Structure paper
Title | Mutation of CDK7 at a conserved residue identifies a common mechanism of acquired resistance to CDK inhibitors in cancer |
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Journal, issue, pages | To Be Published |
Publish date | Nov 27, 2024 (structure data deposition date) |
![]() | Lai C-F / Cushing VI / Bevan CL / Coombes RC / Greber BJ / Buluwela L / Ali S |
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Methods | EM (single particle) |
Resolution | 2.3 - 2.6 Å |
Structure data | EMDB-52205, PDB-9hix: EMDB-52206, PDB-9hiy: EMDB-52207, PDB-9hj0: |
Chemicals | ![]() ChemComp-V0G: ![]() ChemComp-HOH: ![]() ChemComp-AGS: ![]() ChemComp-MG: ![]() ChemComp-I74: |
Source |
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![]() | TRANSFERASE / Kinase / complex / heterotrimer |