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-Structure paper
Title | Discovery of a Novel Series of CHK1 Kinase Inhibitors with Distinctive Hinge Binding Mode |
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Journal, issue, pages | ACS MED. CHEM. LETT., Year 2012 |
Publish date | Oct 19, 2011 (structure data deposition date) |
Authors | Huang, X. / Cheng, C.C. / Fischmann, T.O. / Duca, J.S. / Yang, X. / Richards, M. / Shipps Jr., G.W. |
External links | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.85 Å |
Structure data | PDB-3u9n: |
Chemicals | ChemComp-09H: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / Protein kinase domain / ATPase / ATP Binding / TRANSFERASE-TRANSFERASE INHIBITOR complex |