タイトル | Acetolactate Synthase from Klebsiella pneumoniae in Complex with Mechanism-Based Inhibitor |
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ジャーナル・号・ページ | To Be Published |
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掲載日 | 2015年8月12日 (構造データの登録日) |
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著者 | Latta, A.J. / Andrews, F.H. / McLeish, M.J. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 2.12 - 2.276 Å |
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構造データ | PDB-5d6r: Acetolactate Synthase from Klebsiella pneumoniae in Complex with Mechanism-Based Inhibitor 手法: X-RAY DIFFRACTION / 解像度: 2.276 Å PDB-5wdg: Acetolactate Synthase from Klebsiella pneumoniae in Complex with a Reaction Intermediate 手法: X-RAY DIFFRACTION / 解像度: 2.12 Å |
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化合物 | ChemComp-EN0: 3-[(4-amino-2-methylpyrimidin-5-yl)methyl]-2-[(Z)-2-fluoro-1-hydroxy-2-phosphonoethenyl]-5-(2-{[(S)-hydroxy(phosphonooxy)phosphoryl]oxy}ethyl)-4-methyl-1,3-thiazol-3-ium
ChemComp-A4Y: (2S,3S)-2,3-dihydroxy-3-[(7S,8R,9aS)-8-(2-{[(R)-hydroxy(phosphonooxy)phosphoryl]oxy}ethyl)-2,7-dimethyl-5,7,8,10-tetrahydro-9aH-pyrimido[4,5-d][1,3]thiazolo[3,2-a]pyrimidin-9a-yl]-2-methylbutanoic acid
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由来 | klebsiella pneumoniae (肺炎桿菌)
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キーワード | TRANSFERASE / Inhibition Intermediate Synthase / Intermediate / Synthase / ThDP |
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