+Search query
-Structure paper
Title | Complexes of HIV-1 reverse transcriptase with inhibitors of the HEPT series reveal conformational changes relevant to the design of potent non-nucleoside inhibitors. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 39, Page 1589-1600, Year 1996 |
Publish date | Mar 16, 1996 (structure data deposition date) |
![]() | Hopkins, A.L. / Ren, J. / Esnouf, R.M. / Willcox, B.E. / Jones, E.Y. / Ross, C. / Miyasaka, T. / Walker, R.T. / Tanaka, H. / Stammers, D.K. / Stuart, D.I. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.55 Å |
Structure data | ![]() PDB-1rt1: ![]() PDB-1rt2: |
Chemicals | ![]() ChemComp-MKC: ![]() ChemComp-HOH: ![]() ChemComp-TNK: |
Source |
|
![]() | NUCLEOTIDYLTRANSFERASE / HIV-1 REVERSE TRANSCRIPTASE |