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| Title | Structural basis for asymmetric bis-intercalator targeting of DNA triplex junctions enabling dual inhibition of topoisomerase I and oncogene transcription. |
|---|---|
| Journal, issue, pages | Nucleic Acids Res., Vol. 54, Year 2026 |
| Publish date | May 29, 2025 (structure data deposition date) |
Authors | Wang, S.C. / Hsieh, C.C. / Yuan, T.C. / Lin, S.M. / Chen, C.W. / Chang, C.C. / Huang, S.C. / Wang, E.C. / Huang, Y.J. / Chiang, M.H. ...Wang, S.C. / Hsieh, C.C. / Yuan, T.C. / Lin, S.M. / Chen, C.W. / Chang, C.C. / Huang, S.C. / Wang, E.C. / Huang, Y.J. / Chiang, M.H. / Horng, Y.C. / Hou, M.H. |
External links | Nucleic Acids Res. / PubMed:42206361 |
| Methods | X-ray diffraction |
| Resolution | 1.27 - 1.92 Å |
| Structure data | ![]() PDB-9v87: ![]() PDB-9v88: ![]() PDB-9v89: |
| Chemicals | ![]() ChemComp-SPK: ![]() ChemComp-CO: ![]() ChemComp-CL: ![]() ChemComp-HOH: ![]() ChemComp-ACT: ![]()
ChemComp-XAU: ![]() ChemComp-CA: ![]()
ChemComp-W1H: ![]() ChemComp-MPD: |
| Source |
|
Keywords | DNA / DNA perfectly matched / Watson and Crick base pairing / Ligand-DNA complex / Asymmetric intercalator / Bis-intercalation / Quinoxaline / Acridine |
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