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| Title | Discovery of Zilucoplan: A Complement C5 Inhibitor for Treatment of Anti-Acetylcholine Receptor (AChR) Antibody-Positive Generalized Myasthenia Gravis (gMG). |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 68, Page 25772-25782, Year 2025 |
| Publish date | Sep 8, 2025 (structure data deposition date) |
Authors | Ye, P. / Hammer, R.P. / Wang, Z. / Dhamnaskar, K. / Hoarty, M. / Ma, Z. / Tang, G.Q. / DeMarco, S.J. / Ricardo, A. |
External links | J. Med. Chem. / PubMed:41379101 |
| Methods | X-ray diffraction |
| Resolution | 2 Å |
| Structure data | ![]() PDB-9y6c: |
| Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-8VH: ![]() ChemComp-HOH: |
| Source |
|
Keywords | IMMUNE SYSTEM / Complement / C5 / macrocyclic peptide / Myasthenia Gravis |
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