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| Title | Development of Keap1-Nrf2 Protein-Protein Interaction Inhibitor Activating Intracellular Nrf2 Based on the Naphthalene-2-acetamide Scaffold, and its Anti-Inflammatory Effects. |
|---|---|
| Journal, issue, pages | Chemmedchem, Vol. 20, Page e202500474-e202500474, Year 2025 |
| Publish date | Apr 25, 2025 (structure data deposition date) |
Authors | Yasuda, D. / Toyoshima, K. / Kojima, K. / Ishida, H. / Kaitoh, K. / Imamura, R. / Kanamitsu, K. / Kojima, H. / Funakoshi-Tago, M. / Osawa, M. ...Yasuda, D. / Toyoshima, K. / Kojima, K. / Ishida, H. / Kaitoh, K. / Imamura, R. / Kanamitsu, K. / Kojima, H. / Funakoshi-Tago, M. / Osawa, M. / Ohe, T. / Hirano, T. |
External links | Chemmedchem / PubMed:40902199 |
| Methods | X-ray diffraction |
| Resolution | 1.8 Å |
| Structure data | ![]() PDB-9uo8: |
| Chemicals | ![]() PDB-1l9d: ![]() ChemComp-FMT: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSCRIPTION / PEPTIDE BINDING PROTEIN |
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