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| Title | A Concise and Modular Approach to Generate Novel ROR gamma Agonists. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 68, Page 15849-15871, Year 2025 |
| Publish date | Jul 1, 2025 (structure data deposition date) |
Authors | Fukuda, S. / Ikenogami, T. / Otake, K. / Miwa, S. / Maeda, K. / Yamashita, T. / Inami, T. / Yokota, M. / Lu, Y. / Suma, A. ...Fukuda, S. / Ikenogami, T. / Otake, K. / Miwa, S. / Maeda, K. / Yamashita, T. / Inami, T. / Yokota, M. / Lu, Y. / Suma, A. / Hirono, Y. / Ogawa, N. / Inoue, T. / Harada, K. / Yamaguchi, K. / Akai, S. / Nomura, A. / Adachi, T. / Terawaki, T. / Suzukawa, A. / Kitamoto, M. / Tanimoto, M. / Noguchi, T. / Hata, T. / Kawahara, I. / Iwamoto, K. / Kondo, K. / Kitagawa, Y. / Naka, Y. / Crowe, P. / Tao, H. / Fenn, M. / Thacher, S. / Oba, M. / Shiozaki, M. |
External links | J. Med. Chem. / PubMed:40677142 |
| Methods | X-ray diffraction |
| Resolution | 1.93 Å |
| Structure data | ![]() PDB-9vnx: |
| Chemicals | ![]() PDB-1mam: ![]() ChemComp-EDO: ![]() ChemComp-ACT: ![]() ChemComp-HOH: |
| Source |
|
Keywords | NUCLEAR PROTEIN / nuclear receptor / agonist |
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