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| Title | A long-lasting PI3K delta inhibitor zandelisib forms a water-shielded hydrogen bond with p110 delta and demonstrates sustained inhibitory effects. |
|---|---|
| Journal, issue, pages | Am J Cancer Res, Vol. 15, Page 2097-2110, Year 2025 |
| Publish date | Dec 19, 2024 (structure data deposition date) |
Authors | Kunieda, K. / Nagiri, C. / Watanabe, M. / Yoshida, T. / Zou, J. / Kaneda, A. / Takahashi, Y. / Aburai, K. / Saito, J.I. / Umehara, H. ...Kunieda, K. / Nagiri, C. / Watanabe, M. / Yoshida, T. / Zou, J. / Kaneda, A. / Takahashi, Y. / Aburai, K. / Saito, J.I. / Umehara, H. / Otsu, Y. / Ishii, T. |
External links | Am J Cancer Res / PubMed:40520883 |
| Methods | X-ray diffraction |
| Resolution | 2.5 Å |
| Structure data | ![]() PDB-9l3r: |
| Chemicals | ![]() PDB-1l62: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE/INHIBITOR / Inhibitor / TRANSFERASE / TRANSFERASE-INHIBITOR complex |
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homo sapiens (human)
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