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-Structure paper
| Title | Structure-Guided Design of Affinity/Covalent-Bond Dual-Driven Inhibitors Targeting the AMP Site of FBPase. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 67, Page 20421-20437, Year 2024 |
| Publish date | Dec 6, 2023 (structure data deposition date) |
Authors | Cao, H. / Huang, Z. / Liu, Z. / Zhang, X. / Ren, Y. / Hameed, M.S. / Rao, L. / Makunga, N.P. / Dobrikov, G.M. / Wan, J. |
External links | J. Med. Chem. / PubMed:39520680 |
| Methods | X-ray diffraction |
| Resolution | 2.42 Å |
| Structure data | ![]() PDB-8xbk: |
| Chemicals | ![]()
ChemComp-YR9: ![]() ChemComp-EDO: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
| Source |
|
Keywords | PROTEIN BINDING / covalent inhibitor |
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