+Search query
-Structure paper
Title | A Small-Molecule Inhibitor of Factor Inhibiting HIF Binding to a Tyrosine-flip Pocket for the Treatment of Obesity. |
---|---|
Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Page e202410438-e202410438, Year 2024 |
Publish date | Feb 24, 2023 (structure data deposition date) |
![]() | Wu, Y. / Chen, Y. / Corner, T. / Nakashima, Y. / Salah, E. / Li, Z. / Zhang, L. / Yang, L. / Tumber, A. / Sun, Z. ...Wu, Y. / Chen, Y. / Corner, T. / Nakashima, Y. / Salah, E. / Li, Z. / Zhang, L. / Yang, L. / Tumber, A. / Sun, Z. / Wen, Y. / Zhong, A. / Yang, F. / Li, X. / Zhang, Z. / Schofield, C. / Zhang, X. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.04 - 2.22 Å |
Structure data | ![]() PDB-8ihz: ![]() PDB-8ii0: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-ZN: ![]()
ChemComp-P1X: ![]() ChemComp-HOH: ![]()
ChemComp-P5I: ![]() ChemComp-GOL: |
Source |
|
![]() | OXIDOREDUCTASE / factor-inhibiting hypoxia-inducible factor / FIH / 2OG dependent dioxygenase |