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-Structure paper
Title | Structure-guided conversion from an anaplastic lymphoma kinase inhibitor into Plasmodium lysyl-tRNA synthetase selective inhibitors. |
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Journal, issue, pages | Commun Biol, Vol. 7, Page 742-742, Year 2024 |
Publish date | Aug 1, 2023 (structure data deposition date) |
![]() | Zhou, J. / Xia, M. / Huang, Z. / Qiao, H. / Yang, G. / Qian, Y. / Li, P. / Zhang, Z. / Gao, X. / Jiang, L. ...Zhou, J. / Xia, M. / Huang, Z. / Qiao, H. / Yang, G. / Qian, Y. / Li, P. / Zhang, Z. / Gao, X. / Jiang, L. / Wang, J. / Li, W. / Fang, P. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.92 - 2.83 Å |
Structure data | ![]() PDB-8k9s: ![]() PDB-8k9u: ![]() PDB-8k9v: ![]() PDB-8k9w: ![]() PDB-8k9x: |
Chemicals | ![]() ChemComp-LYS: ![]()
ChemComp-JRU: ![]() ChemComp-MES: ![]() ChemComp-HOH: ![]()
ChemComp-JSL: ![]()
ChemComp-JT4: ![]() ChemComp-GOL: ![]()
ChemComp-JTR: ![]()
ChemComp-JUA: |
Source |
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![]() | LIGASE / lysyl-tRNA synthetase |