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Structure paper

TitleWhat doesn't fit is made to fit: Pim-1 kinase adapts to the configuration of stilbene-based inhibitors.
Journal, issue, pagesArch Pharm, Vol. 357, Page e2400094-e2400094, Year 2024
Publish dateNov 1, 2023 (structure data deposition date)
AuthorsHochban, P.M.M. / Heyder, L. / Heine, A. / Diederich, W.E.
External linksArch Pharm / PubMed:38631036
MethodsX-ray diffraction
Resolution1.89 - 2.45 Å
Structure data

PDB-8r10:
Pim1 in complex with 4-(4-hydroxystyryl)benzoic acid and Pimtide
Method: X-RAY DIFFRACTION / Resolution: 2.2 Å

PDB-8r18:
Pim1 in complex with (E)-4-(4-hydroxystyryl)benzoic acid and Pimtide
Method: X-RAY DIFFRACTION / Resolution: 1.89 Å

PDB-8r1n:
Pim1 in complex with 4-(4-hydroxyphenethyl)benzoic acid and Pimtide
Method: X-RAY DIFFRACTION / Resolution: 2.21 Å

PDB-8r1p:
Pim1 in complex with 6-bromobenzo[d]oxazol-2-amine and Pimtide
Method: X-RAY DIFFRACTION / Resolution: 2.45 Å

PDB-8r1t:
Pim1 in complex with 4-(4-aminophenethyl)benzoic acid and Pimtide
Method: X-RAY DIFFRACTION / Resolution: 2 Å

Chemicals


ChemComp, No image

ChemComp-XGQ:
Unknown entry

ChemComp-HOH:
WATER

ChemComp-GOL:
GLYCEROL


ChemComp, No image

ChemComp-XGK:
Unknown entry

ChemComp-EDO:
1,2-ETHANEDIOL


ChemComp, No image

ChemComp-XIT:
Unknown entry


ChemComp, No image

ChemComp-XIP:
Unknown entry


ChemComp, No image

ChemComp-XIJ:
Unknown entry

Source
  • homo sapiens (human)
KeywordsTRANSFERASE / SERINE KINASE / KINASE / COMPLEX / PIM1 / PIM / PIM-1 / INHIBITOR / TUMORIGENISIS / CANCER / PIMTIDE / PROTO ONCOGEN / ATP / PHOSPHORYLATION / APOPTOSIS / CELL CYCLE

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