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-Structure paper
Title | Structural Analysis of the Macrocyclic Inhibitor BI-4020 Binding to EGFR Kinase. |
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Journal, issue, pages | Chemmedchem, Page e202300343-e202300343, Year 2024 |
Publish date | Dec 6, 2020 (structure data deposition date) |
![]() | Beyett, T.S. / Rana, J.K. / Schaeffner, I.K. / Heppner, D.E. / Eck, M.J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 - 3.1 Å |
Structure data | ![]() PDB-7kxz: ![]() PDB-7ky0: |
Chemicals | ![]() ChemComp-CL: ![]() ChemComp-XA4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / EGFR / kinase / inhibitor / macrocycle / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |