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-Structure paper
Title | A structure-based designed small molecule depletes hRpn13 Pru and a select group of KEN box proteins. |
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Journal, issue, pages | Nat Commun, Vol. 15, Page 2485-2485, Year 2024 |
Publish date | Jan 13, 2023 (structure data deposition date) |
Authors | Lu, X. / Chandravanshi, M. / Sabbasani, V.R. / Gaikwad, S. / Hughitt, V.K. / Gyabaah-Kessie, N. / Scroggins, B.T. / Das, S. / Myint, W. / Clapp, M.E. ...Lu, X. / Chandravanshi, M. / Sabbasani, V.R. / Gaikwad, S. / Hughitt, V.K. / Gyabaah-Kessie, N. / Scroggins, B.T. / Das, S. / Myint, W. / Clapp, M.E. / Schwieters, C.D. / Dyba, M.A. / Bolhuis, D.L. / Koscielniak, J.W. / Andresson, T. / Emanuele, M.J. / Brown, N.G. / Matsuo, H. / Chari, R. / Citrin, D.E. / Mock, B.A. / Swenson, R.E. / Walters, K.J. |
External links | Nat Commun / PubMed:38509117 |
Methods | X-ray diffraction |
Resolution | 2.1 Å |
Structure data | PDB-8ftq: |
Chemicals |
ChemComp-ZTO: ChemComp-HOH: |
Source |
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Keywords | PROTEIN BINDING / Proteasome / Rpn13 / PROTAC |