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-Structure paper
Title | Development of a Series of Pyrrolopyridone MAT2A Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 67, Page 4541-4559, Year 2024 |
Publish date | Aug 30, 2023 (structure data deposition date) |
![]() | Atkinson, S.J. / Bagal, S.K. / Argyrou, A. / Askin, S. / Cheung, T. / Chiarparin, E. / Coen, M. / Collie, I.T. / Dale, I.L. / De Fusco, C. ...Atkinson, S.J. / Bagal, S.K. / Argyrou, A. / Askin, S. / Cheung, T. / Chiarparin, E. / Coen, M. / Collie, I.T. / Dale, I.L. / De Fusco, C. / Dillman, K. / Evans, L. / Feron, L.J. / Foster, A.J. / Grondine, M. / Kantae, V. / Lamont, G.M. / Lamont, S. / Lynch, J.T. / Nilsson Lill, S. / Robb, G.R. / Saeh, J. / Schimpl, M. / Scott, J.S. / Smith, J. / Srinivasan, B. / Tentarelli, S. / Vazquez-Chantada, M. / Wagner, D. / Walsh, J.J. / Watson, D. / Williamson, B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.089 - 1.19 Å |
Structure data | ![]() PDB-8qdy: ![]() PDB-8qdz: ![]() PDB-8qe0: ![]() PDB-8qe1: ![]() PDB-8qe2: ![]() PDB-8qe3: |
Chemicals | ![]()
ChemComp-U74: ![]() ChemComp-SAM: ![]() ChemComp-HOH: ![]()
ChemComp-U6R: ![]()
ChemComp-U8R: ![]()
ChemComp-U8E: ![]()
ChemComp-U7X: ![]()
ChemComp-U96: |
Source |
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![]() | TRANSFERASE / S-Adenosylmethionine biosynthesis / allosteric inhibitor |