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| Title | Identification of small-molecule binding sites of a ubiquitin-conjugating enzyme-UBE2T through fragment-based screening. |
|---|---|
| Journal, issue, pages | Protein Sci., Vol. 33, Page e4904-e4904, Year 2024 |
| Publish date | Jun 26, 2023 (structure data deposition date) |
Authors | Loh, Y.Y. / Anantharajan, J. / Huang, Q. / Xu, W. / Fulwood, J. / Ng, H.Q. / Ng, E.Y. / Gea, C.Y. / Choong, M.L. / Tan, Q.W. ...Loh, Y.Y. / Anantharajan, J. / Huang, Q. / Xu, W. / Fulwood, J. / Ng, H.Q. / Ng, E.Y. / Gea, C.Y. / Choong, M.L. / Tan, Q.W. / Koh, X. / Lim, W.H. / Nacro, K. / Cherian, J. / Baburajendran, N. / Ke, Z. / Kang, C. |
External links | Protein Sci. / PubMed:38358126 |
| Methods | X-ray diffraction |
| Resolution | 1.54 - 1.696 Å |
| Structure data | ![]() PDB-8juc: ![]() PDB-8jvd: |
| Chemicals | ![]()
ChemComp-V23: ![]() ChemComp-EDO: ![]() ChemComp-HOH: ![]()
ChemComp-V2R: |
| Source |
|
Keywords | LIGASE / UBE2T; ubiquitination; fragment-based drug discovery |
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