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TitleDiscovery of TP0628103: A Highly Potent and Selective MMP-7 Inhibitor with Reduced OATP-Mediated Clearance Designed by Shifting Isoelectric Points.
Journal, issue, pagesJ. Med. Chem., Vol. 67, Page 1406-1420, Year 2024
Publish dateJul 20, 2023 (structure data deposition date)
AuthorsOka, Y. / Abe-Sato, K. / Tabuse, H. / Yasukawa, Y. / Yahara, T. / Nishimoto, T. / Kamitani, M. / Fukunaga, T. / Ochiai, N. / Kumasaka-Abe, T. ...Oka, Y. / Abe-Sato, K. / Tabuse, H. / Yasukawa, Y. / Yahara, T. / Nishimoto, T. / Kamitani, M. / Fukunaga, T. / Ochiai, N. / Kumasaka-Abe, T. / Hitaka, K. / Gunji, E. / Ohara, H. / Takeda, T. / Kojima, N. / Asami, T.
External linksJ. Med. Chem. / PubMed:38214909
MethodsX-ray diffraction
Resolution1.7 Å
Structure data

PDB-8k4z:
Crystal structure of human MMP-7 in complex with inhibitor
Method: X-RAY DIFFRACTION / Resolution: 1.7 Å

Chemicals

ChemComp-CA:
Unknown entry

ChemComp-ZN:
Unknown entry

ChemComp-IOD:
IODIDE ION

ChemComp-CL:
Unknown entry

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
  • synthetic construct (others)
KeywordsHYDROLASE / Matrilysin / Matrin / Matrix metalloproteinase-7 / Pump-1 protease / Uterine metalloproteinase

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