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TitleDiscovery and SAR of JTE-151: A Novel ROR gamma Inhibitor for Clinical Development.
Journal, issue, pagesJ. Med. Chem., Vol. 67, Page 952-970, Year 2024
Publish dateNov 24, 2023 (structure data deposition date)
AuthorsMaeba, T. / Hirata, K. / Kotoku, M. / Seki, N. / Maeda, K. / Hirashima, S. / Yamanaka, H. / Sakai, T. / Obika, S. / Hori, A. ...Maeba, T. / Hirata, K. / Kotoku, M. / Seki, N. / Maeda, K. / Hirashima, S. / Yamanaka, H. / Sakai, T. / Obika, S. / Hori, A. / Hara, Y. / Noji, S. / Suwa, Y. / Yokota, M. / Fujioka, S. / Yamaguchi, T. / Katsuda, Y. / Hata, T. / Miyagawa, N. / Arita, K. / Nomura, Y. / Taniguchi, T. / Asahina, K. / Aratsu, Y. / Naka, Y. / Adachi, T. / Nomura, A. / Akai, S. / Oshida, S.I. / Pai, S. / Crowe, P. / Bradley, E. / Steensma, R. / Tao, H. / Fenn, M. / Babine, R. / Li, X. / Thacher, S. / Soeta, T. / Ukaji, Y. / Shiozaki, M.
External linksJ. Med. Chem. / PubMed:38170624
MethodsX-ray diffraction
Resolution2.3 Å
Structure data

PDB-8x7e:
Crystal Structure of the mutant Human ROR gamma Ligand Binding Domain With JTE-151
Method: X-RAY DIFFRACTION / Resolution: 2.3 Å

Chemicals


ChemComp, No image

ChemComp-YAL:
Unknown entry

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsNUCLEAR PROTEIN/INHIBITOR / nuclear receptor / nuclear protein-inhibitor complex

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