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-Structure paper
Title | The discovery of aryl-2-nitroethyl triamino pyrimidines as anti-Trypanosoma brucei agents. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 264, Page 115946-115946, Year 2023 |
Publish date | Mar 13, 2023 (structure data deposition date) |
![]() | Linciano, P. / Pozzi, C. / Tassone, G. / Landi, G. / Mangani, S. / Santucci, M. / Luciani, R. / Ferrari, S. / Santarem, N. / Tagliazucchi, L. ...Linciano, P. / Pozzi, C. / Tassone, G. / Landi, G. / Mangani, S. / Santucci, M. / Luciani, R. / Ferrari, S. / Santarem, N. / Tagliazucchi, L. / Cordeiro-da-Silva, A. / Tonelli, M. / Tondi, D. / Bertarini, L. / Gul, S. / Witt, G. / Moraes, C.B. / Costantino, L. / Costi, M.P. |
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Methods | X-ray diffraction |
Resolution | 1.48 Å |
Structure data | ![]() PDB-8of2: |
Chemicals | ![]() ChemComp-3AY: ![]() ChemComp-NDP: ![]() ChemComp-EDO: ![]() ChemComp-ACT: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / Trypanosoma brucei / pteridine reductase / PTR1 / TbPTR1 / triamminopyrimidine |