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-Structure paper
Title | Identification of Small Molecule Inhibitors and Ligand Directed Degraders of Calcium/Calmodulin Dependent Protein Kinase Kinase 1 and 2 (CaMKK1/2). |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 15750-15760, Year 2023 |
Publish date | Aug 16, 2023 (structure data deposition date) |
![]() | Chen, Y. / Whitefield, B. / Nevius, E. / Hill, M. / DelRosario, J. / Sinitsyna, N. / Shanmugasundaram, V. / Mukherjee, D. / Shi, L. / Mayne, C.G. ...Chen, Y. / Whitefield, B. / Nevius, E. / Hill, M. / DelRosario, J. / Sinitsyna, N. / Shanmugasundaram, V. / Mukherjee, D. / Shi, L. / Mayne, C.G. / Rousseau, A.M. / Bernard, S.M. / Buenviaje, J. / Khambatta, G. / El Samin, M. / Wallace, M. / Nie, Z. / Sivakumar, P. / Hamann, L.G. / McDonnell, D.P. / D'Agostino, L.A. |
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Methods | X-ray diffraction |
Resolution | 1.5 Å |
Structure data | ![]() PDB-8tuc: |
Chemicals | ![]() ChemComp-O7I: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / Calcium/Calmodulin Dependent Protein Kinase Kinase 2 / CAMKK2 / Inhibitor / TRANSFERASE / TRANSFERASE-INHIBITOR complex |