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-Structure paper
Title | Mutate and Conjugate: A Method to Enable Rapid In-Cell Target Validation. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 18, Page 2405-2417, Year 2023 |
Publish date | Feb 15, 2023 (structure data deposition date) |
Authors | Thomas, A.M. / Serafini, M. / Grant, E.K. / Coombs, E.A.J. / Bluck, J.P. / Schiedel, M. / McDonough, M.A. / Reynolds, J.K. / Lee, B. / Platt, M. ...Thomas, A.M. / Serafini, M. / Grant, E.K. / Coombs, E.A.J. / Bluck, J.P. / Schiedel, M. / McDonough, M.A. / Reynolds, J.K. / Lee, B. / Platt, M. / Sharlandjieva, V. / Biggin, P.C. / Duarte, F. / Milne, T.A. / Bush, J.T. / Conway, S.J. |
External links | Acs Chem. Biol. / PubMed:37874862 |
Methods | X-ray diffraction |
Resolution | 1.88 Å |
Structure data | PDB-8ckf: |
Chemicals | ChemComp-E5Q: ChemComp-V0R: ChemComp-HOH: |
Source |
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Keywords | GENE REGULATION / BROMODOMAIN / LIGAND / EPIGENETICS / READER DOMAIN / TRANSCRIPTION REGULATION |