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Title | Structure-Based Optimization and Biological Evaluation of Potent and Selective MMP-7 Inhibitors for Kidney Fibrosis. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 14653-14668, Year 2023 |
Publish date | Jun 26, 2023 (structure data deposition date) |
![]() | Abe-Sato, K. / Tabuse, H. / Kanazawa, H. / Kamitani, M. / Endo, M. / Tokura, S. / Wakabayashi, S. / Yahara, T. / Takeda, T. / Hitaka, K. ...Abe-Sato, K. / Tabuse, H. / Kanazawa, H. / Kamitani, M. / Endo, M. / Tokura, S. / Wakabayashi, S. / Yahara, T. / Takeda, T. / Hitaka, K. / Gunji, E. / Kojima, N. / Oka, Y. |
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Methods | X-ray diffraction |
Resolution | 1.3 - 1.5 Å |
Structure data | ![]() PDB-8jud: ![]() PDB-8juf: ![]() PDB-8jug: |
Chemicals | ![]() ChemComp-CA: ![]() ChemComp-ZN: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / Matrilysin / Matrin / Matrix metalloproteinase-7 / Pump-1 protease / Uterine metalloproteinase / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR complex |