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-Structure paper
タイトル | Calpeptin is a potent cathepsin inhibitor and drug candidate for SARS-CoV-2 infections. |
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ジャーナル・号・ページ | Commun Biol, Vol. 6, Page 1058-1058, Year 2023 |
掲載日 | 2021年12月10日 (構造データの登録日) |
著者 | Reinke, P.Y.A. / de Souza, E.E. / Gunther, S. / Falke, S. / Lieske, J. / Ewert, W. / Loboda, J. / Herrmann, A. / Rahmani Mashhour, A. / Karnicar, K. ...Reinke, P.Y.A. / de Souza, E.E. / Gunther, S. / Falke, S. / Lieske, J. / Ewert, W. / Loboda, J. / Herrmann, A. / Rahmani Mashhour, A. / Karnicar, K. / Usenik, A. / Lindic, N. / Sekirnik, A. / Botosso, V.F. / Santelli, G.M.M. / Kapronezai, J. / de Araujo, M.V. / Silva-Pereira, T.T. / Filho, A.F.S. / Tavares, M.S. / Florez-Alvarez, L. / de Oliveira, D.B.L. / Durigon, E.L. / Giaretta, P.R. / Heinemann, M.B. / Hauser, M. / Seychell, B. / Bohler, H. / Rut, W. / Drag, M. / Beck, T. / Cox, R. / Chapman, H.N. / Betzel, C. / Brehm, W. / Hinrichs, W. / Ebert, G. / Latham, S.L. / Guimaraes, A.M.S. / Turk, D. / Wrenger, C. / Meents, A. |
リンク | Commun Biol / PubMed:37853179 |
手法 | X線回折 |
解像度 | 1.3 - 2 Å |
構造データ | PDB-7qgw: PDB-7qka: PDB-7qkb: PDB-7qkc: PDB-7z3t: PDB-7z3u: PDB-7z58: PDB-8c3d: |
化合物 | ChemComp-CL: ChemComp-MPD: ChemComp-GOL: ChemComp-RN2: ChemComp-HOH: ChemComp-DMS: ChemComp-UED: ChemComp-PEG: ChemComp-NA: ChemComp-PGE: ChemComp-PG4: ChemComp-P6G: ChemComp-EDO: ChemComp-1PE: ChemComp-CA: |
由来 |
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キーワード | HYDROLASE / cathepsin / inhibitor / main protease / MPro / cystein protease / drug development / drug target / peptide-like inhibitor / SARS-CoV-2 / COVID-19 / lysosome / protein degradation / spike protein maturation |