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-Structure paper
Title | Cellular Validation of a Chemically Improved Inhibitor Identifies Monoubiquitination on OTUB2. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 18, Page 2003-2013, Year 2023 |
Publish date | Feb 21, 2023 (structure data deposition date) |
Authors | Gan, J. / de Vries, J. / Akkermans, J.J.L.L. / Mohammed, Y. / Tjokrodirijo, R.T.N. / de Ru, A.H. / Kim, R.Q. / Vargas, D.A. / Pol, V. / Fasan, R. ...Gan, J. / de Vries, J. / Akkermans, J.J.L.L. / Mohammed, Y. / Tjokrodirijo, R.T.N. / de Ru, A.H. / Kim, R.Q. / Vargas, D.A. / Pol, V. / Fasan, R. / van Veelen, P.A. / Neefjes, J. / van Dam, H. / Ovaa, H. / Sapmaz, A. / Geurink, P.P. |
External links | Acs Chem. Biol. / PubMed:37642399 |
Methods | X-ray diffraction |
Resolution | 1.77 Å |
Structure data | PDB-8cms: |
Chemicals | ChemComp-V2X: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / Chemical modification / ubiquitin / deubiquitinase / inhibitor |