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Title | Small molecule branched-chain ketoacid dehydrogenase kinase (BDK) inhibitors with opposing effects on BDK protein levels. |
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Journal, issue, pages | Nat Commun, Vol. 14, Page 4812-4812, Year 2023 |
Publish date | Nov 14, 2022 (structure data deposition date) |
Authors | Roth Flach, R.J. / Bollinger, E. / Reyes, A.R. / Laforest, B. / Kormos, B.L. / Liu, S. / Reese, M.R. / Martinez Alsina, L.A. / Buzon, L. / Zhang, Y. ...Roth Flach, R.J. / Bollinger, E. / Reyes, A.R. / Laforest, B. / Kormos, B.L. / Liu, S. / Reese, M.R. / Martinez Alsina, L.A. / Buzon, L. / Zhang, Y. / Bechle, B. / Rosado, A. / Sahasrabudhe, P.V. / Knafels, J. / Bhattacharya, S.K. / Omoto, K. / Stansfield, J.C. / Hurley, L.D. / Song, L. / Luo, L. / Breitkopf, S.B. / Monetti, M. / Cunio, T. / Tierney, B. / Geoly, F.J. / Delmore, J. / Siddall, C.P. / Xue, L. / Yip, K.N. / Kalgutkar, A.S. / Miller, R.A. / Zhang, B.B. / Filipski, K.J. |
External links | Nat Commun / PubMed:37558654 |
Methods | X-ray diffraction |
Resolution | 2.545 - 3.149 Å |
Structure data | PDB-8f5f: PDB-8f5j: PDB-8f5s: |
Chemicals | ChemComp-ADP: ChemComp-MG: ChemComp-XGG: ChemComp-SO4: ChemComp-HOH: ChemComp-K: ChemComp-XER: ChemComp-XGT: |
Source |
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Keywords | SIGNALING PROTEIN / TRANSFERASE/INHIBITOR / branched chain ketoacid dehydrogenase kinase / inhibitor / TRANSFERASE-INHIBITOR complex |