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-Structure paper
Title | Discovery and Optimization of a STING Agonist Platform for Application in Antibody Drug Conjugates. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 10715-10733, Year 2023 |
Publish date | May 10, 2023 (structure data deposition date) |
![]() | Duvall, J.R. / Thomas, J.D. / Bukhalid, R.A. / Catcott, K.C. / Bentley, K.W. / Collins, S.D. / Eitas, T. / Jones, B.D. / Kelleher, E.W. / Lancaster, K. ...Duvall, J.R. / Thomas, J.D. / Bukhalid, R.A. / Catcott, K.C. / Bentley, K.W. / Collins, S.D. / Eitas, T. / Jones, B.D. / Kelleher, E.W. / Lancaster, K. / Protopopova, M. / Ray, S.S. / Ter-Ovanesyan, E. / Xu, L. / Yang, L. / Zurita, J. / Damelin, M. / Toader, D. / Lowinger, T.B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.72 - 1.97 Å |
Structure data | ![]() PDB-8sth: ![]() PDB-8sti: |
Chemicals | ![]() ChemComp-WWU: ![]() ChemComp-HOH: ![]() ChemComp-WX8: |
Source |
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![]() | IMMUNE SYSTEM/AGONIST / Agonist / STING / IMMUNE SYSTEM / IMMUNE SYSTEM-AGONIST complex |