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-Structure paper
Title | Novel N -(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the beta-Catenin Armadillo Repeats Domain as an Anticancer Agent. |
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Journal, issue, pages | Acs Pharmacol Transl Sci, Vol. 6, Page 1087-1103, Year 2023 |
Publish date | May 4, 2022 (structure data deposition date) |
![]() | Nalli, M. / Di Magno, L. / Wen, Y. / Liu, X. / D'Ambrosio, M. / Puxeddu, M. / Parisi, A. / Sebastiani, J. / Sorato, A. / Coluccia, A. ...Nalli, M. / Di Magno, L. / Wen, Y. / Liu, X. / D'Ambrosio, M. / Puxeddu, M. / Parisi, A. / Sebastiani, J. / Sorato, A. / Coluccia, A. / Ripa, S. / Di Pastena, F. / Capelli, D. / Montanari, R. / Masci, D. / Urbani, A. / Naro, C. / Sette, C. / Orlando, V. / D'Angelo, S. / Biagioni, S. / Bigogno, C. / Dondio, G. / Pastore, A. / Stornaiuolo, M. / Canettieri, G. / Liu, T. / Silvestri, R. / La Regina, G. |
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Methods | X-ray diffraction |
Resolution | 3.434 Å |
Structure data | ![]() PDB-7zrb: |
Chemicals | ![]() ChemComp-JKI: ![]() ChemComp-HOH: |
Source |
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![]() | CELL ADHESION / beta-catenin / colon cancer / wnt pathway |