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-Structure paper
Title | Rational Design of RNA Demethylase FTO Inhibitors with Enhanced Antileukemia Drug-Like Properties. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 9731-9752, Year 2023 |
Publish date | Mar 22, 2023 (structure data deposition date) |
![]() | Xiao, P. / Duan, Z. / Liu, Z. / Chen, L. / Zhang, D. / Liu, L. / Zhou, C. / Gan, J. / Dong, Z. / Yang, C.G. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.14 Å |
Structure data | ![]() PDB-8it9: |
Chemicals | ![]()
ChemComp-ZL6: ![]() ChemComp-AKG: ![]() ChemComp-HOH: |
Source |
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![]() | PROTEIN BINDING / RNA demethylase / RNA binding protein |