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Title | Targeting the Alternative Vitamin E Metabolite Binding Site Enables Noncanonical PPAR gamma Modulation. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 145, Page 14802-14810, Year 2023 |
Publish date | Aug 24, 2022 (structure data deposition date) |
![]() | Arifi, S. / Marschner, J.A. / Pollinger, J. / Isigkeit, L. / Heitel, P. / Kaiser, A. / Obeser, L. / Hofner, G. / Proschak, E. / Knapp, S. ...Arifi, S. / Marschner, J.A. / Pollinger, J. / Isigkeit, L. / Heitel, P. / Kaiser, A. / Obeser, L. / Hofner, G. / Proschak, E. / Knapp, S. / Chaikuad, A. / Heering, J. / Merk, D. |
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Methods | X-ray diffraction |
Resolution | 1.9 - 2.4 Å |
Structure data | ![]() PDB-8aty: ![]() PDB-8atz: ![]() PDB-8cph: ![]() PDB-8cpi: ![]() PDB-8cpj: |
Chemicals | ![]() ChemComp-O7O: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-O86: ![]() ChemComp-WY1: ![]() ChemComp-EDO: |
Source |
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![]() | NUCLEAR PROTEIN / Nuclear receptor / PPARG / inhibitor / Structural Genomics / Structural Genomics Consortium / SGC / DNA BINDING PROTEIN / allosteric inhibitor / orthosteric inhibitor |