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Title | Discovery and Structure-Based Design of Inhibitors of the WD Repeat-Containing Protein 5 (WDR5)-MYC Interaction. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 8310-8323, Year 2023 |
Publish date | Feb 7, 2023 (structure data deposition date) |
![]() | Ding, J. / Liu, L. / Chiang, Y.L. / Zhao, M. / Liu, H. / Yang, F. / Shen, L. / Lin, Y. / Deng, H. / Gao, J. ...Ding, J. / Liu, L. / Chiang, Y.L. / Zhao, M. / Liu, H. / Yang, F. / Shen, L. / Lin, Y. / Deng, H. / Gao, J. / Sage, D.R. / West, L. / Llamas, L.A. / Hao, X. / Kawatkar, S. / Li, E. / Jain, R.K. / Tallarico, J.A. / Canham, S.M. / Wang, H. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.33 - 1.8 Å |
Structure data | ![]() PDB-8g3c: ![]() PDB-8g3e: |
Chemicals | ![]() ChemComp-YJN: ![]() ChemComp-HOH: ![]() ChemComp-YJR: |
Source |
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![]() | ONCOPROTEIN/INHIBITOR / WDR5 / WBM / MYC / small molecule / ONCOPROTEIN-INHIBITOR complex |