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Title | Synthesis and Development of Highly Selective Pyrrolo[2,3- d ]pyrimidine CSF1R Inhibitors Targeting the Autoinhibited Form. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 6959-6980, Year 2023 |
Publish date | Feb 3, 2023 (structure data deposition date) |
![]() | Aarhus, T.I. / Bjornstad, F. / Wolowczyk, C. / Larsen, K.U. / Rognstad, L. / Leithaug, T. / Unger, A. / Habenberger, P. / Wolf, A. / Bjorkoy, G. ...Aarhus, T.I. / Bjornstad, F. / Wolowczyk, C. / Larsen, K.U. / Rognstad, L. / Leithaug, T. / Unger, A. / Habenberger, P. / Wolf, A. / Bjorkoy, G. / Pridans, C. / Eickhoff, J. / Klebl, B. / Hoff, B.H. / Sundby, E. |
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Methods | X-ray diffraction |
Resolution | 1.925 Å |
Structure data | ![]() PDB-8cgc: |
Chemicals | ![]() ChemComp-LMR: ![]() ChemComp-GOL: ![]() ChemComp-UIK: ![]() ChemComp-HOH: |
Source |
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![]() | LIGASE / Kinase / CSF1R / Inhibitors |