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-Structure paper
Title | Application of an "inhalation by design" approach to the identification and in-vitro evaluation of novel purine based PI3K delta inhibitors. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 254, Page 115331-115331, Year 2023 |
Publish date | Oct 17, 2022 (structure data deposition date) |
Authors | Mazzucato, R. / Roberti, M. / Capelli, A.M. / Rancati, F. / Biagetti, M. / Fiorelli, C. / Bruno, P. / Ronchi, P. / Bertolini, S. / Corsi, M. / Pala, D. |
External links | Eur. J. Med. Chem. / PubMed:37094451 |
Methods | X-ray diffraction |
Resolution | 2.43 Å |
Structure data | PDB-8bcy: |
Chemicals | ChemComp-I3H: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / PI3KDELTA KINASE / PI3KDELTA KINASE INHIBITOR |