+Search query
-Structure paper
Title | Discovery of an In Vivo Chemical Probe for BCL6 Inhibition by Optimization of Tricyclic Quinolinones. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 66, Page 5892-5906, Year 2023 |
Publish date | Jan 13, 2023 (structure data deposition date) |
![]() | Harnden, A.C. / Davis, O.A. / Box, G.M. / Hayes, A. / Johnson, L.D. / Henley, A.T. / de Haven Brandon, A.K. / Valenti, M. / Cheung, K.J. / Brennan, A. ...Harnden, A.C. / Davis, O.A. / Box, G.M. / Hayes, A. / Johnson, L.D. / Henley, A.T. / de Haven Brandon, A.K. / Valenti, M. / Cheung, K.J. / Brennan, A. / Huckvale, R. / Pierrat, O.A. / Talbot, R. / Bright, M.D. / Akpinar, H.A. / Miller, D.S.J. / Tarantino, D. / Gowan, S. / de Klerk, S. / McAndrew, P.C. / Le Bihan, Y.V. / Meniconi, M. / Burke, R. / Kirkin, V. / van Montfort, R.L.M. / Raynaud, F.I. / Rossanese, O.W. / Bellenie, B.R. / Hoelder, S. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-8c78: |
Chemicals | ![]() ChemComp-TWI: ![]() ChemComp-EDO: ![]() ChemComp-CL: ![]() ChemComp-HOH: |
Source |
|
![]() | TRANSCRIPTION / Inhibitor / Cancer / Lymphoma |