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-Structure paper
Title | Structure and RAF family kinase isoform selectivity of type II RAF inhibitors tovorafenib and naporafenib. |
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Journal, issue, pages | J. Biol. Chem., Vol. 299, Page 104634-104634, Year 2023 |
Publish date | Nov 20, 2022 (structure data deposition date) |
![]() | Tkacik, E. / Li, K. / Gonzalez-Del Pino, G. / Ha, B.H. / Vinals, J. / Park, E. / Beyett, T.S. / Eck, M.J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.74 - 3.54 Å |
Structure data | ![]() PDB-8f7o: ![]() PDB-8f7p: |
Chemicals | ![]() ChemComp-QOP: ![]() ChemComp-K81: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/INHIBITOR / BRAF / TAK580 / tovorafenib / TRANSFERASE / TRANSFERASE-INHIBITOR complex / LXH254 / naporafenib |