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TitleOxazolo[5,4-f]quinoxaline-type selective inhibitors of glycogen synthase kinase-3 alpha (GSK-3 alpha ): Development and impact on temozolomide treatment of glioblastoma cells.
Journal, issue, pagesBioorg. Chem., Vol. 134, Page 106456-106456, Year 2023
Publish dateAug 26, 2022 (structure data deposition date)
AuthorsHasyeoui, M. / Lassagne, F. / Erb, W. / Nael, M. / Elokely, K.M. / Chaikuad, A. / Knapp, S. / Jorda, A. / Valles, S.L. / Quissac, E. ...Hasyeoui, M. / Lassagne, F. / Erb, W. / Nael, M. / Elokely, K.M. / Chaikuad, A. / Knapp, S. / Jorda, A. / Valles, S.L. / Quissac, E. / Verreault, M. / Robert, T. / Bach, S. / Samarat, A. / Mongin, F.
External linksBioorg. Chem. / PubMed:36913879
MethodsX-ray diffraction
Resolution2.15 - 2.66 Å
Structure data

PDB-8auz:
Crystal structure of GSK3 beta (GSK3b) in complex with FL291.
Method: X-RAY DIFFRACTION / Resolution: 2.66 Å

PDB-8av1:
Crystal structure of GSK3 beta (GSK3b) in complex with CD7.
Method: X-RAY DIFFRACTION / Resolution: 2.15 Å

Chemicals

ChemComp-SO4:
SULFATE ION

ChemComp-O9C:
8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline

ChemComp-HOH:
WATER

ChemComp-EDO:
1,2-ETHANEDIOL

ChemComp-O9L:
2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline

Source
  • homo sapiens (human)
KeywordsTRANSFERASE / kinase / GSK3B / inhibitor / Structural Genomics / Structural Genomics Consortium / SGC

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