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Title | Design, synthesis and characterisation of a novel type II B-RAF paradox breaker inhibitor. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 250, Page 115231-115231, Year 2023 |
Publish date | Jan 17, 2023 (structure data deposition date) |
![]() | Arora, R. / Linders, J.T.M. / Aci-Seche, S. / Verheyen, T. / Van Heerde, E. / Brehmer, D. / Chaikuad, A. / Knapp, S. / Bonnet, P. |
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Methods | X-ray diffraction |
Resolution | 1.65 Å |
Structure data | ![]() PDB-8c7x: ![]() PDB-8c7y: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-BR: ![]() ChemComp-TXV: ![]() ChemComp-HOH: ![]() ChemComp-NO3: |
Source |
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![]() | TRANSFERASE / BRAF / kinase / kinase inhibitor / Structural Genomics / Structural Genomics Consortium / SGC |