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-Structure paper
Title | Discovery of Potent DYRK2 Inhibitors with High Selectivity, Great Solubility, and Excellent Safety Properties for the Treatment of Prostate Cancer. |
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Journal, issue, pages | J. Med. Chem., Vol. 66, Page 4215-4230, Year 2023 |
Publish date | Dec 1, 2022 (structure data deposition date) |
![]() | Yuan, K. / Shen, H. / Zheng, M. / Xia, F. / Li, Q. / Chen, W. / Ji, M. / Yang, H. / Zhuang, X. / Cai, Z. ...Yuan, K. / Shen, H. / Zheng, M. / Xia, F. / Li, Q. / Chen, W. / Ji, M. / Yang, H. / Zhuang, X. / Cai, Z. / Min, W. / Wang, X. / Xiao, Y. / Yang, P. |
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Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | ![]() PDB-8hlt: |
Chemicals | ![]() ChemComp-XSE: |
Source |
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![]() | CELL CYCLE / Inhibitor |