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-Structure paper
Title | 2-Ethynylbenzaldehyde-Based, Lysine-Targeting Irreversible Covalent Inhibitors for Protein Kinases and Nonkinases. |
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Journal, issue, pages | J. Am. Chem. Soc., Year 2023 |
Publish date | Oct 19, 2022 (structure data deposition date) |
Authors | Chen, P. / Tang, G. / Zhu, C. / Sun, J. / Wang, X. / Xiang, M. / Huang, H. / Wang, W. / Li, L. / Zhang, Z.M. ...Chen, P. / Tang, G. / Zhu, C. / Sun, J. / Wang, X. / Xiang, M. / Huang, H. / Wang, W. / Li, L. / Zhang, Z.M. / Gao, L. / Yao, S.Q. |
External links | J. Am. Chem. Soc. / PubMed:36774655 |
Methods | X-ray diffraction |
Resolution | 1.4640844632 - 2.4501342407 Å |
Structure data | PDB-8h7b: PDB-8h7f: PDB-8h7h: |
Chemicals | ChemComp-QHR: ChemComp-HOH: ChemComp-QEW: ChemComp-QH9: |
Source |
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Keywords | TRANSFERASE / Complex / inhibitor / lysine |