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-Structure paper
Title | A novel pan-selective bromodomain inhibitor for epigenetic drug design. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 249, Page 115139-115139, Year 2023 |
Publish date | Nov 25, 2020 (structure data deposition date) |
Authors | Warstat, R. / Pervaiz, M. / Regenass, P. / Amann, M. / Schmidtkunz, K. / Einsle, O. / Jung, M. / Breit, B. / Hugle, M. / Gunther, S. |
External links | Eur. J. Med. Chem. / PubMed:36736153 |
Methods | X-ray diffraction |
Resolution | 1.92 Å |
Structure data | PDB-7b1t: |
Chemicals | ChemComp-SOK: ChemComp-DMS: ChemComp-HOH: |
Source |
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Keywords | PROTEIN BINDING / BRD4 / BRD4(1) / BET / MPM6 / Bromodomain / inhibitor / co-crystal / cocrystal / fragment |