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-Structure paper
Title | Nutlin-3a-aa: Improving the Bioactivity of a p53/MDM2 Interaction Inhibitor by Introducing a Solvent-Exposed Methylene Group. |
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Journal, issue, pages | Chembiochem, Vol. 24, Page e202300006-e202300006, Year 2023 |
Publish date | Jul 13, 2022 (structure data deposition date) |
Authors | Nietzold, F. / Rubner, S. / Labuzek, B. / Golik, P. / Surmiak, E. / Del Corte, X. / Kitel, R. / Protzel, C. / Reppich-Sacher, R. / Stichel, J. ...Nietzold, F. / Rubner, S. / Labuzek, B. / Golik, P. / Surmiak, E. / Del Corte, X. / Kitel, R. / Protzel, C. / Reppich-Sacher, R. / Stichel, J. / Magiera-Mularz, K. / Holak, T.A. / Berg, T. |
External links | Chembiochem / PubMed:36602436 |
Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | PDB-8aeu: |
Chemicals | ChemComp-BME: ChemComp-M0L: ChemComp-HOH: |
Source |
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Keywords | LIGASE / Biological activity / drug design / inhibitors / protein-protein interactions |