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-Structure paper
Title | Targeting BRD4 and PI3K signaling pathways for the treatment of medulloblastoma. |
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Journal, issue, pages | J Control Release, Vol. 354, Page 80-90, Year 2023 |
Publish date | Apr 25, 2022 (structure data deposition date) |
![]() | Sethi, B. / Kumar, V. / Jayasinghe, T.D. / Dong, Y. / Ronning, D.R. / Zhong, H.A. / Coulter, D.W. / Mahato, R.I. |
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Methods | X-ray diffraction |
Resolution | 1.2 - 2.5 Å |
Structure data | ![]() PDB-7usg: ![]() PDB-7ush: ![]() PDB-7usi: ![]() PDB-7usj: ![]() PDB-7usk: |
Chemicals | ![]() ChemComp-O6O: ![]() ChemComp-EDO: ![]() ChemComp-NA: ![]() ChemComp-HOH: ![]() ChemComp-82V: ![]() ChemComp-PEG: ![]() ChemComp-DMS: ![]() ChemComp-CL: ![]() ChemComp-PGE: |
Source |
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![]() | TRANSCRIPTION/INHIBITOR / Inhibitor / acetyllysine binding pocket / TRANSCRIPTION / TRANSCRIPTION-INHIBITOR complex / TRANSCRIPTON/INHIBITOR / TRANSCRIPTON-INHIBITOR complex |