Structures of a constitutively active mutant of human IDH3 reveal new insights into the mechanisms of allosteric activation and the catalytic reaction.
PDB-8grb: Crystal structure of a constitutively active mutant of the alpha beta heterodimer of human IDH3 手法: X-RAY DIFFRACTION / 解像度: 2.848 Å
PDB-8grd: Crystal structure of a constitutively active mutant of the alpha beta heterodimer of human IDH3 in complex with ADP and Mg 手法: X-RAY DIFFRACTION / 解像度: 2.699 Å
PDB-8grg: Crystal structure of a constitutively active mutant of the alpha gamma heterodimer of human IDH3 手法: X-RAY DIFFRACTION / 解像度: 2.699 Å
PDB-8grh: Crystal structure of a constitutively active mutant of the alpha gamma heterodimer of human IDH3 in complex with CIT 手法: X-RAY DIFFRACTION / 解像度: 2.506 Å
PDB-8gru: Crystal structure of a constitutively active mutant of the alpha beta heterodimer of human IDH3 in complex with ICT, NAD and Ca 手法: X-RAY DIFFRACTION / 解像度: 2.847 Å
PDB-8gs5: Crystal structure of a constitutively active mutant of human IDH3 holoenzyme in apo form 手法: X-RAY DIFFRACTION / 解像度: 4.486 Å