+Search query
-Structure paper
Title | Rational design of the zonulin inhibitor AT1001 derivatives as potential anti SARS-CoV-2. |
---|---|
Journal, issue, pages | Eur. J. Med. Chem., Vol. 244, Page 114857-114857, Year 2022 |
Publish date | May 13, 2022 (structure data deposition date) |
Authors | Di Micco, S. / Rahimova, R. / Sala, M. / Scala, M.C. / Vivenzio, G. / Musella, S. / Andrei, G. / Remans, K. / Mammri, L. / Snoeck, R. ...Di Micco, S. / Rahimova, R. / Sala, M. / Scala, M.C. / Vivenzio, G. / Musella, S. / Andrei, G. / Remans, K. / Mammri, L. / Snoeck, R. / Bifulco, G. / Di Matteo, F. / Vestuto, V. / Campiglia, P. / Marquez, J.A. / Fasano, A. |
External links | Eur. J. Med. Chem. / PubMed:36332548 |
Methods | X-ray diffraction |
Resolution | 1.336 - 1.999 Å |
Structure data | PDB-7zv5: PDB-7zv7: PDB-7zv8: |
Chemicals | ChemComp-DMS: ChemComp-HOH: ChemComp-OCA: |
Source |
|
Keywords | ANTIVIRAL PROTEIN / SARS Cov-2 / 3CL / main protease |