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-Structure paper
Title | Structure-Based Design of Active-Site-Directed, Highly Potent, Selective, and Orally Bioavailable Low-Molecular-Weight Protein Tyrosine Phosphatase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 13892-13909, Year 2022 |
Publish date | May 2, 2022 (structure data deposition date) |
![]() | He, R. / Wang, J. / Yu, Z.H. / Moyers, J.S. / Michael, M.D. / Durham, T.B. / Cramer, J.W. / Qian, Y. / Lin, A. / Wu, L. ...He, R. / Wang, J. / Yu, Z.H. / Moyers, J.S. / Michael, M.D. / Durham, T.B. / Cramer, J.W. / Qian, Y. / Lin, A. / Wu, L. / Noinaj, N. / Barrett, D.G. / Zhang, Z.Y. |
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Methods | X-ray diffraction |
Resolution | 1.5 Å |
Structure data | ![]() PDB-7uw6: |
Chemicals | ![]() ChemComp-OIF: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / low molecular weight protein tyrosine phosphatase; Inhibitor; Complex |