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-Structure paper
| Title | Promising antimalarials targeting apicoplast DNA polymerase from Plasmodium falciparum. |
|---|---|
| Journal, issue, pages | Eur. J. Med. Chem., Vol. 243, Page 114751-114751, Year 2022 |
| Publish date | Nov 23, 2021 (structure data deposition date) |
Authors | Chheda, P.R. / Nieto, N. / Kaur, S. / Beck, J.M. / Beck, J.R. / Honzatko, R. / Kerns, R.J. / Nelson, S.W. |
External links | Eur. J. Med. Chem. / PubMed:36191407 |
| Methods | X-ray diffraction |
| Resolution | 2.5 - 2.7 Å |
| Structure data | ![]() PDB-7sxl: ![]() PDB-7sxq: |
| Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-NA: ![]() ChemComp-CL: ![]() ChemComp-PEG: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
| Source |
|
Keywords | REPLICATION / Transferase / DNA polymerase / exonulease / apicoplast / Plasmodium falciparum |
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