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Title | Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1 alpha ,25-Dihydroxyvitamin D 3. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 13112-13124, Year 2022 |
Publish date | Apr 1, 2022 (structure data deposition date) |
Authors | Seoane, S. / Gogoi, P. / Zarate-Ruiz, A. / Peluso-Iltis, C. / Peters, S. / Guiberteau, T. / Maestro, M.A. / Perez-Fernandez, R. / Rochel, N. / Mourino, A. |
External links | J. Med. Chem. / PubMed:36166643 |
Methods | X-ray diffraction |
Resolution | 2.6 - 2.62 Å |
Structure data | PDB-7zfg: PDB-7zfx: |
Chemicals | ChemComp-ACT: ChemComp-IV5: ChemComp-HOH: ChemComp-IV1: |
Source |
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Keywords | TRANSCRIPTION / complex / agonist / vitamin D receptor |