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-Structure paper
Title | GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A 2A Adenosine Receptor. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 11648-11657, Year 2022 |
Publish date | May 16, 2022 (structure data deposition date) |
![]() | Shiriaeva, A. / Park, D. / Kim, G. / Lee, Y. / Hou, X. / Jarhad, D.B. / Yu, J. / Hyun, Y.E. / Kim, W. / Gao, Z.G. ...Shiriaeva, A. / Park, D. / Kim, G. / Lee, Y. / Hou, X. / Jarhad, D.B. / Yu, J. / Hyun, Y.E. / Kim, W. / Gao, Z.G. / Jacobson, K.A. / Han, G.W. / Stevens, R.C. / Jeong, L.S. / Choi, S. / Cherezov, V. |
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Methods | X-ray diffraction |
Resolution | 2.05 - 2.8 Å |
Structure data | ![]() PDB-8cu6: ![]() PDB-8cu7: |
Chemicals | ![]() ChemComp-OLA: ![]() ChemComp-OLC: ![]() ChemComp-PEG: ![]() ChemComp-LJX: ![]() ChemComp-CLR: ![]() ChemComp-HOH: ![]() ChemComp-NA: ![]() ChemComp-ETF: |
Source |
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![]() | MEMBRANE PROTEIN / GPCR / A2a adenosine receptor / LCP / nucleoside / antagonist / molecular dynamics / S277A mutant |