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-Structure paper
Title | Discovery of the First Selective Nanomolar Inhibitors of ERAP2 by Kinetic Target-Guided Synthesis. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 61, Page e202203560-e202203560, Year 2022 |
Publish date | Oct 7, 2021 (structure data deposition date) |
Authors | Camberlein, V. / Fleau, C. / Sierocki, P. / Li, L. / Gealageas, R. / Bosc, D. / Guillaume, V. / Warenghem, S. / Leroux, F. / Rosell, M. ...Camberlein, V. / Fleau, C. / Sierocki, P. / Li, L. / Gealageas, R. / Bosc, D. / Guillaume, V. / Warenghem, S. / Leroux, F. / Rosell, M. / Cheng, K. / Medve, L. / Prigent, M. / Decanter, M. / Piveteau, C. / Biela, A. / Eveque, M. / Dumont, J. / Mpakali, A. / Giastas, P. / Herledan, A. / Couturier, C. / Haupenthal, J. / Lesire, L. / Hirsch, A.K.H. / Deprez, B. / Stratikos, E. / Bouvier, M. / Deprez-Poulain, R. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:35904863 |
Methods | X-ray diffraction |
Resolution | 3.2 Å |
Structure data | PDB-7sh0: |
Chemicals | ChemComp-ZN: ChemComp-GIY: ChemComp-EPE: ChemComp-MES: ChemComp-NA: ChemComp-HOH: |
Source |
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Keywords | IMMUNE SYSTEM / HYDROLASE/INHIBITOR / AMINOPEPTIDASE / ERAP2 STRUCTURE / ENZYME INHIBITOR / ANTIGEN PROCESSING / HYDROLASE-INHIBITOR complex |