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-Structure paper
Title | Interaction of CYP3A4 with Rationally Designed Ritonavir Analogues: Impact of Steric Constraints Imposed on the Heme-Ligating Group and the End-Pyridine Attachment. |
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Journal, issue, pages | Int J Mol Sci, Vol. 23, Year 2022 |
Publish date | Mar 22, 2022 (structure data deposition date) |
![]() | Samuels, E.R. / Sevrioukova, I.F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.25 - 2.9 Å |
Structure data | ![]() PDB-7uf9: ![]() PDB-7ufa: ![]() PDB-7ufb: ![]() PDB-7ufc: ![]() PDB-7ufd: ![]() PDB-7ufe: ![]() PDB-7uff: |
Chemicals | ![]() ChemComp-HEM: ![]() ChemComp-NH0: ![]() ChemComp-NI6: ![]() ChemComp-HOH: ![]() ChemComp-NJ0: ![]() ChemComp-NJO: ![]() ChemComp-T0K: ![]() ChemComp-GOL: ![]() ChemComp-NXR: ![]() ChemComp-PO4: ![]() ChemComp-NYF: |
Source |
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![]() | OXIDOREDUCTASE/INHIBITOR / CYP3A4 / inhibitor / complex / OXIDOREDUCTASE / OXIDOREDUCTASE-INHIBITOR complex |